SCHEMBL28260312

SCHEMBL28260312

COc1ccc(OC)c(Nc2cc(NC(=O)Nc3c(Cl)cccc3Cl)ncn2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 1.00
FGFR1 P11362 4/20 1.00
ERBB3 P21860 4/20 0.61
KDR P35968 2/20 0.56
ABL1 P00519 1/20 0.56
PDGFRB P09619 1/20 0.56
KIT P10721 1/20 0.56
SRC P12931 1/20 0.56
BRAF P15056 1/20 0.56
EPHB4 P54760 1/20 0.56
TEK Q02763 1/20 0.56
FGFR3 P22607 3/20 0.52
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
MAPT P10636 3/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
LCK P06239 1/20 0.47
GAA P10253 2/20 0.47
USP2 O75604 1/20 0.47
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28905573 0.86 EGFR (0.75) EGFRFGFR1ERBB3KDRABL1
SCHEMBL28261624 0.84 EGFR (1.00) EGFRFGFR1ERBB3KDRABL1
SCHEMBL28515074 0.83 EGFR (0.71) EGFRFGFR1ERBB3KDRABL1
SCHEMBL374876 0.83 EGFR (0.71) EGFRFGFR1ERBB3FGFR3MEN1
SCHEMBL28498357 0.79 EGFR (0.66) EGFRFGFR1ERBB3FGFR3MEN1
SCHEMBL28514560 0.77 EGFR (0.64) EGFRFGFR1KDRABL1PDGFRB
SCHEMBL374173 0.77 EGFR (0.75) EGFRFGFR1ERBB3KDRABL1
SCHEMBL28489979 0.76 EGFR (0.62) EGFRFGFR1ERBB3MEN1KMT2A
SCHEMBL28465755 0.75 EGFR (0.65) EGFRFGFR1ERBB3SRCMEN1
SCHEMBL28497440 0.75 EGFR (0.60) EGFRFGFR1ERBB3FGFR3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109053593-B 1- (2, 6-chlorphenyl) -3- (substituted pyrimidine-4-yl) urea compound and preparation and application thereof 温州医科大学 2020-12-04 CN claimed
CN-109053593-A 1- (2,6- chlorphenyl) -3- (substituted pyrimidines -4- base) carbamide compounds and its preparation and application 温州医科大学 2018-12-21 CN claimed
CN-109053593-B 1- (2, 6-chlorphenyl) -3- (substituted pyrimidine-4-yl) urea compound and preparation and application thereof 温州医科大学 2020-12-04 CN disclosed