SCHEMBL28260409

SCHEMBL28260409

C[Si](C)(C)C#Cc1cc([N+](=O)[O-])cnc1Cl

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.40
GAA P10253 1/20 0.40
ALDH1A1 P00352 5/20 0.36
VCAM1 P19320 1/20 0.36
IDO1 P14902 1/20 0.36
GLA P06280 2/20 0.35
AHR P35869 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.33
RECQL P46063 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MAPK1 P28482 1/20 0.33
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1368267 0.82 IDO1 (0.46) HTTGAAALDH1A1IDO1GLA
SCHEMBL28160052 0.79 HTT (0.41) HTTGAAALDH1A1VCAM1IDO1
SCHEMBL30618307 0.78 VCAM1 (0.56) HTTGAAALDH1A1VCAM1GLA
SCHEMBL1816348 0.78 VCAM1 (0.56) HTTGAAALDH1A1VCAM1GLA
SCHEMBL28445576 0.75 CCR1 (0.32) ALDH1A1TDP1
SCHEMBL28452456 0.75 PLAU (0.35) HTTALDH1A1IDO1TDP1HSD17B10
SCHEMBL15544241 0.74 HSD17B10 (0.51) HTTGAAALDH1A1VCAM1MEN1
SCHEMBL30334705 0.74 HSD17B10 (0.51) HTTGAAALDH1A1VCAM1MEN1
SCHEMBL30549997 0.74 ALDH1A1 (0.40) HTTGAAALDH1A1IDO1MEN1
SCHEMBL17629991 0.72 GAA (0.41) HTTGAAALDH1A1VCAM1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109053742-A New tricyclic compound ABBVIE 公司 2018-12-21 CN disclosed