SCHEMBL28260548

SCHEMBL28260548

c1ccc(-c2cc(-c3ccsc3)[nH]c2-c2ccccc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GCGR P47871 2/20 0.52
MAPK14 Q16539 2/20 0.52
CYP2E1 P05181 1/20 0.50
CYP2A6 P11509 1/20 0.50
CYP2B6 P20813 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4793206 0.82 GCGR (0.65) GCGRMAPK14
Piperazine SCHEMBL28060957 0.74 GCGR (0.56) GCGRMAPK14
SCHEMBL28552564 0.72 GCGR (0.61) GCGRMAPK14
SCHEMBL28542916 0.72 GCGR (0.61) GCGRMAPK14
SCHEMBL28154907 0.72 GCGR (0.61) GCGRMAPK14
SCHEMBL28912040 0.72 GCGR (0.82) GCGRMAPK14
SCHEMBL4778800 0.72 GCGR (0.51) GCGRMAPK14
SCHEMBL8987160 0.72 CYP2E1 (0.53) CYP2E1CYP2A6CYP2B6
SCHEMBL7058734 0.72 CYP2A6 (0.70) CYP2E1CYP2A6CYP2B6
SCHEMBL27870289 0.70 CYP2A6 (0.67) CYP2E1CYP2A6CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108863890-B 4-pyrroline-2-ketone derivative and preparation method thereof 厦门华厦学院 2021-04-20 CN disclosed
CN-108863890-A A kind of 4- pyrroline-2-one derivative and preparation method thereof 厦门华厦学院 2018-11-23 CN disclosed