SCHEMBL28264372

SCHEMBL28264372

COC(=O)c1ccc2c(c1)NCCN2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.50
CA2 P00918 3/20 0.50
ALDH1A1 P00352 3/20 0.50
CA12 O43570 2/20 0.50
CA7 P43166 2/20 0.50
CA9 Q16790 2/20 0.50
CA14 Q9ULX7 2/20 0.50
LMNA P02545 2/20 0.50
XDH P47989 1/20 0.50
ALOX5 P09917 1/20 0.48
MAPT P10636 4/20 0.47
HSD17B10 Q99714 4/20 0.46
HPGD P15428 3/20 0.46
KDM4E B2RXH2 3/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
ATM Q13315 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29721687 0.89 CA1 (0.50) CA1CA2ALDH1A1CA12CA7
SCHEMBL288320 0.81 MAPT (0.54) CA1CA2ALDH1A1CA12CA7
SCHEMBL30445913 0.81 MAPT (0.54) CA1CA2ALDH1A1CA12CA7
SCHEMBL2898350 0.81 ALDH1A1 (0.47) CA1CA2ALDH1A1CA12CA7
SCHEMBL29906783 0.81 ALDH1A1 (0.47) CA1CA2ALDH1A1CA12CA7
Hydrochloric Acid SCHEMBL699425 0.80 MAPT (0.53) CA1CA2ALDH1A1CA12CA7
Hydrochloric Acid SCHEMBL3102567 0.80 ALDH1A1 (0.46) CA1CA2ALDH1A1CA12CA7
Hydrochloric Acid SCHEMBL29940234 0.80 ALDH1A1 (0.46) CA1CA2ALDH1A1CA12CA7
SCHEMBL45146 0.79 MAPT (0.68) CA1CA2ALDH1A1CA12CA7
SCHEMBL22226391 0.79 ALDH1A1 (0.51) CA1CA2ALDH1A1CA12CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108997229-B 1,2,3, 4-tetrahydroquinoxaline-6-carboxylic acid methyl ester and preparation method thereof 郑州轻工业学院 2020-05-05 CN claimed
CN-108997229-A 1,2,3,4- tetrahydroquinoxaline -6- carboxylate methyl ester and preparation method thereof 郑州轻工业学院 2018-12-14 CN claimed
CN-108997229-B 1,2,3, 4-tetrahydroquinoxaline-6-carboxylic acid methyl ester and preparation method thereof 郑州轻工业学院 2020-05-05 CN disclosed
CN-108997229-B 1,2,3, 4-tetrahydroquinoxaline-6-carboxylic acid methyl ester and preparation method thereof 郑州轻工业学院 2020-05-05 CN disclosed
CN-108997229-B 1,2,3, 4-tetrahydroquinoxaline-6-carboxylic acid methyl ester and preparation method thereof 郑州轻工业学院 2020-05-05 CN disclosed
CN-110573154-A Compositions and methods for modulating short-chain dehydrogenase activity 卡斯西部储备大学 2019-12-13 CN disclosed
CN-108997229-A 1,2,3,4- tetrahydroquinoxaline -6- carboxylate methyl ester and preparation method thereof 郑州轻工业学院 2018-12-14 CN disclosed
CN-108997229-A 1,2,3,4- tetrahydroquinoxaline -6- carboxylate methyl ester and preparation method thereof 郑州轻工业学院 2018-12-14 CN disclosed
CN-108997229-A 1,2,3,4- tetrahydroquinoxaline -6- carboxylate methyl ester and preparation method thereof 郑州轻工业学院 2018-12-14 CN disclosed