SCHEMBL28264649

SCHEMBL28264649

c1cn(C2CCCCC2)c(-c2ccsc2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.39
HTR6 P50406 2/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
DRD2 P14416 1/20 0.36
HRH4 Q9H3N8 2/20 0.35
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
CCNE1 P24864 2/20 0.35
CDK2 P24941 2/20 0.35
GRM1 Q13255 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27761911 0.78 LMNA (0.43) KDM4EALDH1A1GAAMAPTLMNA
SCHEMBL28400995 0.77 NPC1 (0.40) KDM4EALDH1A1MEN1GAAKMT2A
SCHEMBL28598328 0.73 KDM4E (0.51) KDM4EALDH1A1SMN1; SMN2MEN1GAA
SCHEMBL28598336 0.72 ALDH1A1 (0.38) ALDH1A1MAPTCHRM2CHRM4CHRM5
SCHEMBL28713147 0.71 HPGD (0.43) KDM4EALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL29286631 0.71 ADORA1 (0.41) KMT2AIDO1LMNA
SCHEMBL28226097 0.69 ESR1 (0.41) KDRKDM4EALDH1A1KMT2AMAPT
SCHEMBL28713138 0.69 FLT1 (0.40) KDM4EALDH1A1SMN1; SMN2MEN1GAA
SCHEMBL28695130 0.69 ABL1 (0.51) KDM4EALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL11015922 0.69 KDM4E (0.40) KDM4EGAAGRM1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109096139-B Preparation method of alpha-carbonyl amide derivative 贵州大学 2021-03-02 CN disclosed
CN-110997682-A Inhibitors of indoleamine 2, 3-dioxygenase and/or tryptophan 2, 3-dioxygenase 爱杜西亚药品有限公司 2020-04-10 CN disclosed
CN-109096139-A A kind of preparation method of alpha-carbonyl amide derivatives 贵州大学 2018-12-28 CN disclosed