SCHEMBL28264653

SCHEMBL28264653

COc1ccc(-n2ccnc2-c2cccc(OC)c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.56
NPSR1 Q6W5P4 2/20 0.56
TSHR P16473 2/20 0.56
RAB9A P51151 2/20 0.56
LMNA P02545 1/20 0.56
DYRK1A Q13627 2/20 0.50
CLK4 Q9HAZ1 2/20 0.50
KDR P35968 3/20 0.49
FLT1 P17948 2/20 0.49
FLT4 P35916 2/20 0.49
COMT P21964 1/20 0.48
TP53 P04637 1/20 0.47
THRB P10828 1/20 0.47
GRM1 Q13255 2/20 0.47
TNK2 Q07912 1/20 0.46
ALDH1A1 P00352 2/20 0.46
RXFP1 Q9HBX9 1/20 0.46
MAPK9 P45984 1/20 0.45
MAPK10 P53779 1/20 0.45
PTGS2 P35354 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12077033 0.91 KDR (0.55) MAPTNPSR1TSHRRAB9ALMNA
SCHEMBL28600687 0.89 KMT2A (0.46) MAPTNPSR1TSHRRAB9ALMNA
SCHEMBL11385870 0.87 KDR (0.58) MAPTTSHRRAB9ALMNAKDR
SCHEMBL11771718 0.85 KDR (0.49) RAB9ADYRK1ACLK4KDRTP53
SCHEMBL23382222 0.84 KDR (0.59) MAPTLMNADYRK1ACLK4KDR
SCHEMBL30878105 0.84 KDR (0.59) MAPTLMNADYRK1ACLK4KDR
SCHEMBL15315965 0.83 TUBB4A (0.44) MAPTRAB9ALMNADYRK1ACLK4
SCHEMBL28186197 0.81 KDR (0.55) RAB9ACLK4KDRFLT1FLT4
SCHEMBL3278138 0.81 MAPK9 (0.58) RAB9ADYRK1AKDRTP53MAPK9
SCHEMBL12076906 0.81 KDR (0.50) MAPTNPSR1TSHRRAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109096139-B Preparation method of alpha-carbonyl amide derivative 贵州大学 2021-03-02 CN disclosed
CN-109096139-A A kind of preparation method of alpha-carbonyl amide derivatives 贵州大学 2018-12-28 CN disclosed