SCHEMBL28274307

SCHEMBL28274307

C[C@@H]1CNCCN1.O=COCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
HTR2C P28335 2/20 0.42
LTA4H P09960 1/20 0.41
MAOB P27338 1/20 0.39
GLA P06280 1/20 0.39
HTR2A P28223 1/20 0.38
LMNA P02545 1/20 0.37
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
CYP2C19 P33261 1/20 0.35
HTR1A P08908 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27791206 1.00 TSHR (0.42) TSHRHTR2CLTA4HMAOBGLA
SCHEMBL27939939 1.00 TSHR (0.42) TSHRHTR2CLTA4HMAOBGLA
SCHEMBL28270587 0.84 TSHR (0.46) TSHRHTR2CGLASLC6A2SLC6A4
Piperazine SCHEMBL28083640 0.84 TACR1 (0.42) TSHRHTR2CMAOBHTR2ALMNA
Piperazine SCHEMBL27484195 0.84 TACR1 (0.42) TSHRHTR2CMAOBHTR2ALMNA
SCHEMBL28796114 0.83 LTA4H (0.46) TSHRHTR2CLTA4HMAOBGLA
Piperazine SCHEMBL28258210 0.82 TACR1 (0.41) TSHRHTR2CMAOBHTR2ALMNA
SCHEMBL28139300 0.82 TSHR (0.42) TSHRHTR2CMAOBHTR2ASLC6A2
Azetidine SCHEMBL27976635 0.81 TSHR (0.41) TSHRHTR2CMAOBLMNASLC6A2
SCHEMBL27825232 0.81 TSHR (0.49) TSHRHTR2CLTA4HGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311867-A Conjugate comprising RIPK2 inhibitor 葛兰素史克知识产权开发有限公司 2019-02-05 CN disclosed
CN-105793238-A Substituted benzamides and methods of use thereof 基因泰克公司 2016-07-20 CN disclosed