SCHEMBL28279773

SCHEMBL28279773

Nc1[nH]nc2c1CC(NNC(=O)OCc1ccccc1)CC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.43
CA2 P00918 4/20 0.43
ACHE P22303 2/20 0.43
TSHR P16473 1/20 0.43
ALDH1A1 P00352 2/20 0.42
GAA P10253 1/20 0.42
TLR4 O00206 1/20 0.39
CA12 O43570 2/20 0.39
CA9 Q16790 2/20 0.39
EPHX1 P07099 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
CPB1 P15086 1/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19643187 0.92 CA1 (0.53) CA1CA2ACHETSHRALDH1A1
SCHEMBL19642834 0.92 CA1 (0.53) CA1CA2ACHETSHRALDH1A1
SCHEMBL19642779 0.92 CA1 (0.53) CA1CA2ACHETSHRALDH1A1
SCHEMBL28870334 0.79 CA1 (0.47) CA1CA2ACHETSHRALDH1A1
SCHEMBL22227927 0.72 ALDH1A1 (0.55) CA1CA2ACHETSHRALDH1A1
SCHEMBL21843301 0.71 ALDH1A1 (0.64) CA1CA2TSHRALDH1A1GAA
SCHEMBL22492335 0.70 DHFR (0.54) ALDH1A1GAAMEN1KMT2ACYP2C19
SCHEMBL2170012 0.70 ALDH1A1 (0.67) CA1CA2TSHRALDH1A1GAA
SCHEMBL2169031 0.70 ALDH1A1 (0.67) CA1CA2TSHRALDH1A1GAA
SCHEMBL27787789 0.70 ALDH1A1 (0.54) CA1CA2TSHRALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109475530-A For treating the aminoacyl indazole immunomodulator of autoimmune disease 洛克菲勒大学 2019-03-15 CN disclosed