SCHEMBL28280620

SCHEMBL28280620

NC(=O)c1ccc(N(CCCl)CCCl)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.58
ERBB2 P04626 5/20 0.58
ALDH1A1 P00352 4/20 0.53
CYP3A4 P08684 3/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
HIF1A Q16665 3/20 0.53
LMNA P02545 3/20 0.53
ALOX15 P16050 2/20 0.53
NFKB1 P19838 2/20 0.53
THPO P40225 2/20 0.53
MAPT P10636 2/20 0.53
PMP22 Q01453 2/20 0.53
KMT2A Q03164 2/20 0.53
ABCB11 O95342 1/20 0.53
CHRM2 P08172 1/20 0.53
ADRA2A P08913 1/20 0.53
CHRM1 P11229 1/20 0.53
ACHE P22303 1/20 0.53
PTGS1 P23219 1/20 0.53
OPRM1 P35372 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9163920 0.93 EGFR (0.53) EGFRERBB2ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL9248366 0.83 EGFR (0.47) EGFRERBB2ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL7462603 0.82 EGFR (0.60) EGFRERBB2ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL766052 0.82 EGFR (0.61) EGFRERBB2ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL11980711 0.81 EGFR (0.63) EGFRERBB2ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL2170152 0.80 EGFR (0.54) EGFRERBB2ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL14839588 0.78 CYP3A4 (0.58) EGFRERBB2ALDH1A1CYP3A4SMN1; SMN2
Hydrochloric Acid SCHEMBL10535649 0.78 CYP3A4 (0.50) EGFRERBB2ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL5384052 0.77 CYP3A4 (0.49) EGFRERBB2ALDH1A1CYP3A4SMN1; SMN2
SCHEMBL12266656 0.77 EGFR (0.58) EGFRERBB2ALDH1A1CYP3A4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109574960-A A kind of docetaxel derivative and its preparation method and application 南京友怡医药科技有限公司 2019-04-05 CN claimed
CN-109574960-A A kind of docetaxel derivative and its preparation method and application 南京友怡医药科技有限公司 2019-04-05 CN disclosed