SCHEMBL2828337

SCHEMBL2828337

O=c1ocnn1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.44
ALDH1A1 P00352 7/20 0.42
HTT P42858 5/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
LMNA P02545 3/20 0.42
NPSR1 Q6W5P4 3/20 0.42
NPC1 O15118 2/20 0.42
MAPT P10636 2/20 0.42
RAB9A P51151 2/20 0.42
PAX8 Q06710 2/20 0.42
MITF O75030 1/20 0.42
S1PR4 O95977 1/20 0.42
THRB P10828 1/20 0.42
XBP1 P17861 1/20 0.42
S1PR1 P21453 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
GAA P10253 2/20 0.41
HIF1A Q16665 1/20 0.41
CA9 Q16790 1/20 0.40
CYP2C9 P11712 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10579384 0.80 NPC1 (0.42) POLBSMN1; SMN2LMNANPC1MAPT
SCHEMBL31027122 0.78 NPC1 (0.50) POLBALDH1A1LMNANPC1MAPT
SCHEMBL11884923 0.71 PEPD (0.43) ALDH1A1LMNANPC1MAPTGAA
SCHEMBL8386697 0.70 TDP1 (0.44) POLBALDH1A1HTTLMNAMAPT
SCHEMBL10763332 0.68 GSK3B (0.41) ALDH1A1NPC1RAB9AGAAKDM4E
SCHEMBL14435888 0.68 HTT (0.49) POLBALDH1A1HTTSMN1; SMN2NPC1
SCHEMBL30710827 0.67 CYP1A2 (0.40) ALDH1A1LMNANPSR1MAPTS1PR4
SCHEMBL11249037 0.65 POLB (0.38) POLBALDH1A1HTTSMN1; SMN2LMNA
SCHEMBL13787110 0.64 MGLL (0.45) ALDH1A1HTTLMNACA9KMT2A
SCHEMBL11337998 0.64 MGLL (0.45) ALDH1A1HTTLMNACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118231766-A Application of oxadiazolone compound, electrolyte and preparation method thereof, solid electrolyte membrane, lithium ion battery and electric equipment 比亚迪股份有限公司 2024-06-21 CN claimed
EP-0854871-B1 1,3,4-OXADIAZOLIN-2-ONES AND THEIR USE AS PESTICIDES BAYER AG (DE) 2000-08-16 EP claimed
US-6013804-A FOR CONTROLLING ANIMAL PESTS BAYER AKTIENGESELLSCHAFT (DE) 2000-01-11 US claimed
EP-0854871-A1 1,3,4-OXADIAZOLIN-2-ONES AND THEIR USE AS PESTICIDES BAYER AG (DE) 1998-07-29 EP claimed
WO-1997008158-A1 1,3,4-OXADIAZOLIN-2-ONES AND THEIR USE AS PESTICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-03-06 WO claimed
EP-4562016-A2 CDK2 INHIBITORS AND METHODS OF USING THE SAME Cedilla Therapeutics, Inc. (US) 2025-06-04 EP disclosed
CN-118231766-A Application of oxadiazolone compound, electrolyte and preparation method thereof, solid electrolyte membrane, lithium ion battery and electric equipment 比亚迪股份有限公司 2024-06-21 CN disclosed
WO-2024026483-A2 CDK2 INHIBITORS AND METHODS OF USING THE SAME CEDILLA THERAPEUTICS, INC. (US) 2024-02-01 WO disclosed
EP-2570418-A2 2,3-dihydro-6-nitroimidazo[2,1-b]oxazoles compound OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2013-03-20 EP disclosed
EP-2238131-A1 5-O-SUBSTITUTED 3-N-PHENYL-1,3,4-OXADIAZOLONES FOR MEDICAL USE BIAL - Portela & Ca., S.A. (PT) 2010-10-13 EP disclosed
EP-2238131-A1 5-O-SUBSTITUTED 3-N-PHENYL-1,3,4-OXADIAZOLONES FOR MEDICAL USE BIAL - Portela & Ca., S.A. (PT) 2010-10-13 EP disclosed
EP-2238131-A1 5-O-SUBSTITUTED 3-N-PHENYL-1,3,4-OXADIAZOLONES FOR MEDICAL USE BIAL - Portela & Ca., S.A. (PT) 2010-10-13 EP disclosed
WO-2010074587-A2 5-O-SUBSTITUTED 3-N-ARYL-1,3,4-OXADIAZOLONES FOR MEDICAL USE BIAL - PORTELA & CA., S.A. (PT) 2010-07-01 WO disclosed
WO-2009084970-A1 5-O-SUBSTITUTED 3-N-PHENYL-1,3,4-OXADIAZOLONES FOR MEDICAL USE BIAL-PORTELA & COMPANHIA, S.A. (PT) 2009-07-09 WO disclosed
WO-2009084970-A1 5-O-SUBSTITUTED 3-N-PHENYL-1,3,4-OXADIAZOLONES FOR MEDICAL USE BIAL-PORTELA & COMPANHIA, S.A. (PT) 2009-07-09 WO disclosed
EP-0854871-B1 1,3,4-OXADIAZOLIN-2-ONES AND THEIR USE AS PESTICIDES BAYER AG (DE) 2000-08-16 EP disclosed
US-6013804-A FOR CONTROLLING ANIMAL PESTS BAYER AKTIENGESELLSCHAFT (DE) 2000-01-11 US disclosed
US-5869509-A TREAT DISORDERS RESPONSIVE TO OPENERS OF THE LARGE CONDUCTANCE CALCIUM-ACTIVATED POTASSIUM CHANNELS BRISTOL-MYERS SQUIBB COMPANY (US) 1999-02-09 US disclosed
EP-0854871-A1 1,3,4-OXADIAZOLIN-2-ONES AND THEIR USE AS PESTICIDES BAYER AG (DE) 1998-07-29 EP disclosed
WO-1997008158-A1 1,3,4-OXADIAZOLIN-2-ONES AND THEIR USE AS PESTICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-03-06 WO disclosed