SCHEMBL28286346

SCHEMBL28286346

CNC(=O)c1ccc(Nc2ccncc2C(N)=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 6/20 0.51
SYK P43405 2/20 0.51
MKNK1 Q9BUB5 1/20 0.46
MKNK2 Q9HBH9 1/20 0.46
NUDT1 P36639 1/20 0.45
SIRT3 Q9NTG7 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
JAK2 O60674 3/20 0.43
JAK1 P23458 3/20 0.43
TYK2 P29597 1/20 0.43
PTK2 Q05397 2/20 0.42
TGFBR1 P36897 1/20 0.42
AURKA O14965 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28284462 0.85 SIRT2 (0.54) SIRT2NUDT1SIRT3TDP1JAK2
SCHEMBL5078983 0.83 SIRT3 (0.54) SIRT2SYKSIRT3TDP1TGFBR1
SCHEMBL479807 0.80 SIRT2 (0.54) SIRT2SIRT3TDP1JAK2JAK1
SCHEMBL3569822 0.77 SIRT3 (0.61) SIRT2MKNK1MKNK2SIRT3TDP1
SCHEMBL2714846 0.76 SIRT2 (0.53) SIRT2SIRT3TDP1JAK2JAK1
SCHEMBL2717397 0.74 MAPK9 (0.51) SIRT2SIRT3TDP1TGFBR1
SCHEMBL2717012 0.74 MAPK9 (0.51) SIRT2SIRT3TDP1
SCHEMBL22201589 0.74 IRAK4 (0.54) SIRT3TDP1POLB
SCHEMBL12986577 0.74 TDP1 (0.53) NUDT1SIRT3TDP1TGFBR1POLB
SCHEMBL5083064 0.73 PTGS1 (0.57) SIRT2SYKSIRT3TDP1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109641906-A HETEROARYL SUBSTITUTED AMINOPYRIDINE COMPOUNDS 百时美施贵宝公司 2019-04-16 CN claimed
CN-109641906-A HETEROARYL SUBSTITUTED AMINOPYRIDINE COMPOUNDS 百时美施贵宝公司 2019-04-16 CN disclosed