SCHEMBL28290680

SCHEMBL28290680

NC(=O)c1ccc2c(c1)C=CNN2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.35
PARP1 P09874 8/20 0.35
TSHR P16473 3/20 0.35
PLAU P00749 1/20 0.34
HSD17B10 Q99714 3/20 0.33
ALDH1A1 P00352 2/20 0.33
PARP15 Q460N3 2/20 0.33
PARP14 Q460N5 2/20 0.33
PARP10 Q53GL7 2/20 0.33
KMT2A Q03164 2/20 0.33
PARP16 Q8N5Y8 1/20 0.33
PARP11 Q9NR21 1/20 0.33
PARP4 Q9UKK3 1/20 0.33
TNKS O95271 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
KDM4E B2RXH2 1/20 0.33
BRD4 O60885 1/20 0.33
BRPF1 P55201 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1007936 0.76 LCK (0.37) LCKSIRT2PARP1TSHRPLAU
SCHEMBL17476748 0.73 LCK (0.40) LCKPARP1TSHRHSD17B10ALDH1A1
Hydrochloric Acid SCHEMBL4766162 0.71 LCK (0.39) LCKPARP1TSHRHSD17B10ALDH1A1
SCHEMBL31750688 0.71 TSHR (0.38) LCKSIRT2PARP1TSHRHSD17B10
SCHEMBL27973449 0.71 TSHR (0.38) LCKSIRT2PARP1TSHRHSD17B10
SCHEMBL1227619 0.69 LCK (0.34) LCKSIRT2PARP1TSHRHSD17B10
SCHEMBL12056910 0.69 SIRT2 (0.50) LCKSIRT2PARP1TSHRHSD17B10
SCHEMBL23304599 0.68 PARP1 (0.44) LCKSIRT2PARP1TSHRHSD17B10
SCHEMBL9995986 0.68 TSHR (0.45) LCKPARP1TSHRHSD17B10ALDH1A1
SCHEMBL2357761 0.68 LCK (0.36) LCKPARP1TSHRPLAUHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109575016-A PDE9 inhibitors and uses thereof 南京药捷安康生物科技有限公司 2019-04-05 CN disclosed