SCHEMBL28291327

SCHEMBL28291327

NC(=O)OCC(=O)NC1CCNCC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 3/20 0.50
GNAI3 P08754 1/20 0.46
GNAO1 P09471 1/20 0.46
GNAI1 P63096 1/20 0.46
POLB P06746 3/20 0.46
NPSR1 Q6W5P4 1/20 0.42
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
ATM Q13315 1/20 0.41
CHRM5 P08912 1/20 0.41
CHRM3 P20309 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
USP2 O75604 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
ESR2 Q92731 1/20 0.39
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656762 0.83 EPHX1 (0.50) EPHX1GNAI3GNAO1GNAI1POLB
SCHEMBL4070701 0.80 EPHX1 (0.55) EPHX1GNAI3GNAO1GNAI1POLB
SCHEMBL15447812 0.79 NPSR1 (0.68) EPHX1GNAI3GNAO1GNAI1POLB
SCHEMBL21882064 0.79 EPHX1 (0.53) EPHX1GNAI3GNAO1GNAI1POLB
SCHEMBL13927599 0.78 EPHX1 (0.57) EPHX1GNAI3GNAO1GNAI1POLB
SCHEMBL18872267 0.77 GNAI3 (0.48) EPHX1GNAI3GNAO1GNAI1POLB
SCHEMBL28291418 0.76 GNAI3 (0.44) EPHX1GNAI3GNAO1GNAI1POLB
SCHEMBL31314544 0.76 EPHX1 (0.59) EPHX1GNAI3GNAO1GNAI1POLB
SCHEMBL14676023 0.75 NPSR1 (0.37) POLBNPSR1KMT2AMEN1ATM
SCHEMBL19764243 0.75 GNAI3 (0.49) EPHX1GNAI3GNAO1GNAI1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563043-B Substituted pyridines as inhibitors of DNMT1 葛兰素史密斯克莱知识产权发展有限公司 2022-05-31 CN disclosed
CN-109563043-A SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 葛兰素史密斯克莱知识产权发展有限公司 2019-04-02 CN disclosed