SCHEMBL28291329

SCHEMBL28291329

NC(=O)COc1cccc(F)c1F

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.53
HTT P42858 1/20 0.53
CTSB P07858 1/20 0.45
KCNN4 O15554 1/20 0.45
HPGD P15428 1/20 0.42
CES2 O00748 1/20 0.41
BCHE P06276 1/20 0.41
CES1 P23141 1/20 0.41
GRM2 Q14416 2/20 0.40
LMNA P02545 1/20 0.40
FKBP1A P62942 1/20 0.40
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ADRB2 P07550 1/20 0.39
PARP10 Q53GL7 1/20 0.39
CASP1 P29466 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11212903 0.85 HTT (0.61) KDM4EHTTKCNN4HPGDLMNA
SCHEMBL13696493 0.83 HTT (0.50) KDM4EHTTKCNN4HPGDLMNA
SCHEMBL5362778 0.78 HTT (0.71) KDM4EHTTLMNAPOLBSMN1; SMN2
Trifluoroacetic Acid SCHEMBL23202690 0.77 HTT (0.55) KDM4EHTTKCNN4HPGDLMNA
SCHEMBL28692786 0.76 KMT2A (0.45) KCNN4HPGDCES2BCHECES1
SCHEMBL3949993 0.75 PKM (0.50) KDM4EHTTHPGDLMNAPOLB
SCHEMBL13506327 0.74 LMNA (0.56) KDM4ECES2BCHECES1GRM2
SCHEMBL23112144 0.73 KDM4E (0.59) KDM4EHPGDGRM2SMN1; SMN2
SCHEMBL10436878 0.73 KDM4E (0.64) KDM4EHTTHPGDLMNAPOLB
SCHEMBL5251365 0.73 HTT (0.54) KDM4EHTTHPGDPOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563043-A SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 葛兰素史密斯克莱知识产权发展有限公司 2019-04-02 CN disclosed