SCHEMBL2829134

SCHEMBL2829134

Cc1cc(-c2ccc(C(F)(F)F)cc2)cn2c(-c3nc(-c4cnc(N)nc4)c[nH]3)cnc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.39
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
CDK9 P50750 1/20 0.39
LCK P06239 1/20 0.35
KIT P10721 1/20 0.35
SRC P12931 1/20 0.35
KDR P35968 1/20 0.35
ALOX5AP P20292 9/20 0.34
FEN1 P39748 9/20 0.34
CDK5 Q00535 2/20 0.34
CDK5R1 Q15078 2/20 0.34
NPBWR1 P48145 1/20 0.34
FYN P06241 1/20 0.32
CLK1 P49759 2/20 0.32
ADORA2A P29274 1/20 0.32
MC4R P32245 1/20 0.32
NTRK1 P04629 1/20 0.32
CSF1R P07333 1/20 0.32
NTRK2 Q16620 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2829132 0.82 LCK (0.35) CCNT1CCNA2CDK2CDK9LCK
SCHEMBL313597 0.79 LMNA (0.42) ALOX5AP
SCHEMBL1348445 0.73 LCK (0.38) LCKKITSRCKDRALOX5AP
SCHEMBL313095 0.72 LMNA (0.42) NPBWR1
SCHEMBL1346318 0.71 SCN5A (0.40) SRC
SCHEMBL1349224 0.68 SCN5A (0.37) SRC
SCHEMBL312385 0.67 PTPN11 (0.42)
SCHEMBL312216 0.67 S1PR1 (0.47)
SCHEMBL12111313 0.66 COMT (0.41) NPBWR1CLK1
SCHEMBL1348661 0.66 SCN5A (0.35) SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1934214-B1 OXADIAZOLYL PYRAZOLO-PYRIMIDINES AS MGLUR2 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-04-07 EP claimed