SCHEMBL28291412

SCHEMBL28291412

c1ccc(N2CCNCC2)c(C2CCNCC2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 4/20 0.59
HTR1A P08908 3/20 0.56
SLC6A2 P23975 1/20 0.56
SLC6A4 P31645 1/20 0.56
HTR2C P28335 7/20 0.53
HTR2A P28223 3/20 0.50
HTR6 P50406 3/20 0.50
HTR7 P34969 2/20 0.50
HTR5A P47898 2/20 0.50
DRD2 P14416 2/20 0.50
DRD3 P35462 2/20 0.50
HTR3E A5X5Y0 2/20 0.50
HTR3B O95264 2/20 0.50
HTR3A P46098 2/20 0.50
HTR3D Q70Z44 2/20 0.50
HTR3C Q8WXA8 2/20 0.50
SIGMAR1 Q99720 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
NCF1 P14598 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8291557 0.95 ADRB1 (0.61) ADRB1HTR1ASLC6A2SLC6A4HTR2A
Hydrochloric Acid SCHEMBL7836810 0.93 HTR1A (0.59) ADRB1HTR1ASLC6A2SLC6A4HTR2C
SCHEMBL15834289 0.91 HTR2C (0.51) ADRB1HTR1ASLC6A2SLC6A4HTR2C
SCHEMBL4849498 0.90 ADRB1 (0.56) ADRB1HTR1ASLC6A2SLC6A4HTR2C
SCHEMBL18701462 0.90 HTR2C (0.50) ADRB1HTR1ASLC6A2SLC6A4HTR2C
SCHEMBL4849474 0.90 ADRB1 (0.56) ADRB1HTR1ASLC6A2SLC6A4HTR2C
SCHEMBL4856101 0.90 ADRB1 (0.56) ADRB1HTR1ASLC6A2SLC6A4HTR2C
SCHEMBL27868018 0.87 HTR2C (0.47) ADRB1HTR1ASLC6A2SLC6A4HTR2C
SCHEMBL4420245 0.87 ADRB1 (0.53) ADRB1HTR1ASLC6A2SLC6A4HTR2A
SCHEMBL4258576 0.84 ADRB1 (0.50) ADRB1HTR1ASLC6A2SLC6A4HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563043-A SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 葛兰素史密斯克莱知识产权发展有限公司 2019-04-02 CN disclosed