SCHEMBL28292565

SCHEMBL28292565

O=C(c1ccccn1)N1CCOC[C@H]1CO

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.49
NTRK1 P04629 2/20 0.48
HCRTR1 O43613 13/20 0.44
HCRTR2 O43614 13/20 0.44
CYP3A4 P08684 8/20 0.44
PDK1 Q15118 1/20 0.43
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNA7 P36544 1/20 0.41
CHRNA4 P43681 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17600702 0.80 L3MBTL1 (0.53) L3MBTL1NTRK1CYP3A4CHRNB2CHRNB4
SCHEMBL17600703 0.80 L3MBTL1 (0.53) L3MBTL1NTRK1CYP3A4CHRNB2CHRNB4
SCHEMBL17600727 0.80 PDK1 (0.48) L3MBTL1NTRK1HCRTR1HCRTR2CYP3A4
SCHEMBL17600728 0.80 PDK1 (0.48) L3MBTL1NTRK1HCRTR1HCRTR2CYP3A4
Hydrochloric Acid SCHEMBL17600714 0.79 PDK1 (0.47) L3MBTL1HCRTR1HCRTR2CYP3A4PDK1
SCHEMBL28941055 0.76 NTRK1 (0.41) NTRK1PDK1ALDH1A1SMN1; SMN2
SCHEMBL28941108 0.76 NTRK1 (0.41) NTRK1PDK1ALDH1A1SMN1; SMN2
SCHEMBL28294291 0.76 NTRK1 (0.41) NTRK1PDK1ALDH1A1SMN1; SMN2
SCHEMBL30589306 0.76 SMN1; SMN2 (0.46) HCRTR1HCRTR2CYP3A4PDK1ALDH1A1
SCHEMBL28941054 0.76 SCN9A (0.40) NTRK1HCRTR1HCRTR2PDK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed