SCHEMBL28292572

SCHEMBL28292572

O=C(c1cc[c]cn1)N1CCO[C@@H](CO)C1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 0.44
PDK1 Q15118 3/20 0.42
ALOX5AP P20292 1/20 0.41
FEN1 P39748 1/20 0.41
PIK3CA P42336 2/20 0.41
PIK3CD O00329 1/20 0.40
PIK3R2 O00459 1/20 0.40
PIK3CB P42338 1/20 0.40
PIK3CG P48736 1/20 0.40
PIK3R5 Q8WYR1 1/20 0.40
PIK3R3 Q92569 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
LRRK2 Q5S007 1/20 0.37
KDM1A O60341 1/20 0.35
ROCK2 O75116 1/20 0.35
JAK2 O60674 3/20 0.35
ABL1 P00519 1/20 0.35
RAB9A P51151 2/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3984592 0.81 PDK1 (0.47) SCN9APDK1ALOX5APFEN1PIK3CA
SCHEMBL28292603 0.79 SCN9A (0.48) SCN9APDK1ALOX5APFEN1PIK3CA
SCHEMBL744843 0.77 SMN1; SMN2 (0.57) SMN1; SMN2RAB9A
SCHEMBL22341858 0.75 SCN9A (0.44) SCN9APDK1ALOX5APFEN1PIK3CA
SCHEMBL22341860 0.75 SCN9A (0.44) SCN9APDK1ALOX5APFEN1PIK3CA
SCHEMBL28941104 0.75 SCN9A (0.44) SCN9APDK1ALOX5APFEN1PIK3CA
SCHEMBL28941103 0.74 SCN9A (0.49) SCN9APDK1ALOX5APFEN1PIK3CA
SCHEMBL28941076 0.74 SCN9A (0.49) SCN9APDK1ALOX5APFEN1PIK3CA
SCHEMBL3983890 0.73 CYP19A1 (0.48) PDK1SMN1; SMN2RAB9AKMT2A
SCHEMBL3984591 0.72 PDK1 (0.43) SCN9APDK1ALOX5APFEN1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed