SCHEMBL28292603

SCHEMBL28292603

Nc1ccc(C(=O)N2CCO[C@H](CO)C2)nc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 0.48
ALOX5AP P20292 1/20 0.46
FEN1 P39748 1/20 0.46
PIK3CA P42336 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
KDM5A P29375 1/20 0.43
PIK3CD O00329 1/20 0.43
PIK3R2 O00459 1/20 0.43
PIK3CB P42338 1/20 0.43
PIK3CG P48736 1/20 0.43
PIK3R5 Q8WYR1 1/20 0.43
PIK3R3 Q92569 1/20 0.43
PDK1 Q15118 1/20 0.43
LRRK2 Q5S007 1/20 0.40
CCR8 P51685 5/20 0.39
KCNH2 Q12809 5/20 0.39
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
KDM1A O60341 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28941076 0.82 SCN9A (0.49) SCN9AALOX5APFEN1PIK3CASMN1; SMN2
SCHEMBL28941103 0.82 SCN9A (0.49) SCN9AALOX5APFEN1PIK3CASMN1; SMN2
SCHEMBL13725365 0.82 PDK1 (0.47) SCN9AALOX5APFEN1PIK3CAPIK3CD
SCHEMBL28941104 0.81 SCN9A (0.44) SCN9AALOX5APFEN1PIK3CASMN1; SMN2
SCHEMBL22341858 0.81 SCN9A (0.44) SCN9AALOX5APFEN1PIK3CASMN1; SMN2
SCHEMBL22341860 0.81 SCN9A (0.44) SCN9AALOX5APFEN1PIK3CASMN1; SMN2
SCHEMBL28292572 0.79 SCN9A (0.44) SCN9AALOX5APFEN1PIK3CASMN1; SMN2
SCHEMBL3227298 0.78 SMN1; SMN2 (0.70) SMN1; SMN2CCR8KCNH2
SCHEMBL3232177 0.74 IRAK4 (0.42) SCN9AALOX5APFEN1SMN1; SMN2KDM5A
SCHEMBL15651191 0.74 ADORA2A (0.48) PIK3CASMN1; SMN2PIK3CDPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed