SCHEMBL28292590

SCHEMBL28292590

CC(C)(O)CCOc1ccccn1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.46
CYP2D6 P10635 2/20 0.40
SMN1; SMN2 Q16637 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NPC1 O15118 3/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP2C19 P33261 1/20 0.38
GRM2 Q14416 1/20 0.38
RAB9A P51151 2/20 0.38
MCHR1 Q99705 1/20 0.37
PIM1 P11309 1/20 0.37
GABRA5 P31644 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10202933 0.85 TSHR (0.44) TSHRCYP2D6SMN1; SMN2L3MBTL1NPC1
SCHEMBL14771962 0.81 TSHR (0.48) TSHRCYP2D6SMN1; SMN2L3MBTL1NPC1
SCHEMBL13310631 0.80 TSHR (0.43) TSHRCYP2D6SMN1; SMN2L3MBTL1NPC1
SCHEMBL4190714 0.78 KDM4E (0.50) TSHRCYP2D6SMN1; SMN2L3MBTL1NPC1
SCHEMBL25917658 0.78 TSHR (0.44) TSHRCYP2D6SMN1; SMN2L3MBTL1NPC1
SCHEMBL29608023 0.78 EPHX2 (0.45) TSHRCYP2D6SMN1; SMN2L3MBTL1NPC1
SCHEMBL28028435 0.78 EPHX2 (0.45) TSHRCYP2D6SMN1; SMN2L3MBTL1NPC1
SCHEMBL27890078 0.77 P2RX7 (0.35) CYP2D6ALDH1A1PIM1
SCHEMBL19783211 0.76 CYP2D6 (0.41) CYP2D6ALDH1A1MCHR1PIM1TP53
SCHEMBL2416582 0.75 ALDH1A1 (0.50) TSHRCYP2D6SMN1; SMN2L3MBTL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed