SCHEMBL28292910

SCHEMBL28292910

NS(=O)(=O)c1ccc(-n2nc(C(=O)N3CCSCC3)cc2-c2ccc(Cl)cc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 1.00
CHRNA7 P36544 5/20 0.83
PTGS1 P23219 2/20 0.81
CHRNB2 P17787 1/20 0.72
CHRNA4 P43681 1/20 0.72
MALT1 Q9UDY8 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28294504 0.90 PTGS2 (1.00) PTGS2CHRNA7PTGS1
SCHEMBL28872998 0.90 PTGS2 (1.00) PTGS2CHRNA7PTGS1
SCHEMBL28294503 0.90 PTGS2 (1.00) PTGS2CHRNA7PTGS1
SCHEMBL28294514 0.90 PTGS2 (1.00) PTGS2CHRNA7PTGS1
SCHEMBL28292889 0.89 PTGS2 (1.00) PTGS2CHRNA7PTGS1CHRNB2CHRNA4
SCHEMBL28292993 0.88 PTGS2 (1.00) PTGS2CHRNA7CHRNB2CHRNA4
SCHEMBL28294491 0.87 PTGS2 (1.00) PTGS2CHRNA7PTGS1
SCHEMBL28292908 0.87 PTGS2 (1.00) PTGS2CHRNA7PTGS1
SCHEMBL28294627 0.85 PTGS2 (1.00) PTGS2CHRNA7PTGS1
SCHEMBL28294510 0.83 PTGS2 (1.00) PTGS2CHRNA7PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109748872-A The design and synthesis of the morpholine derivative antitumoral compounds of one kind skeleton containing diaryl pyrazole 南京大学 2019-05-14 CN disclosed