SCHEMBL28292908

SCHEMBL28292908

COc1ccc(-c2cc(C(=O)N3CCSCC3)nn2-c2ccc(S(N)(=O)=O)cc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 1.00
PTGS1 P23219 2/20 0.74
CHRNA7 P36544 2/20 0.67
CA1 P00915 1/20 0.62
CA2 P00918 1/20 0.62
CA9 Q16790 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28292943 0.90 PTGS2 (1.00) PTGS2PTGS1CA1CA2CA9
SCHEMBL28294627 0.90 PTGS2 (1.00) PTGS2PTGS1CHRNA7
SCHEMBL28294504 0.89 PTGS2 (1.00) PTGS2PTGS1CHRNA7CA9
SCHEMBL28292903 0.89 PTGS2 (1.00) PTGS2CHRNA7
SCHEMBL28292910 0.87 PTGS2 (1.00) PTGS2PTGS1CHRNA7
SCHEMBL28872998 0.87 PTGS2 (1.00) PTGS2PTGS1CHRNA7CA1CA2
SCHEMBL28294503 0.87 PTGS2 (1.00) PTGS2PTGS1CHRNA7
SCHEMBL28294514 0.87 PTGS2 (1.00) PTGS2PTGS1CHRNA7
SCHEMBL28294491 0.85 PTGS2 (1.00) PTGS2PTGS1CHRNA7
SCHEMBL6351220 0.83 CHRNA7 (0.78) PTGS2PTGS1CHRNA7CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109748872-A The design and synthesis of the morpholine derivative antitumoral compounds of one kind skeleton containing diaryl pyrazole 南京大学 2019-05-14 CN disclosed