SCHEMBL28292981

SCHEMBL28292981

Clc1cccc2nc(Br)nc(Cl)c12

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.42
ELANE P08246 4/20 0.42
GRIN1 Q05586 4/20 0.39
GRIN2A Q12879 4/20 0.39
ACHE P22303 3/20 0.39
BCHE P06276 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
PBRM1 Q86U86 2/20 0.38
PSMB8 P28062 1/20 0.36
C1R P00736 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30013654 0.79 PARP1 (0.44) PARP1ELANEGRIN1GRIN2AACHE
SCHEMBL3337344 0.79 PARP1 (0.44) PARP1ELANEGRIN1GRIN2AACHE
SCHEMBL7417855 0.76 PARP1 (0.50) PARP1ELANEGRIN1GRIN2AACHE
SCHEMBL18283409 0.74 TDP1 (0.41) PARP1ELANEGRIN1GRIN2AACHE
SCHEMBL9263229 0.73 KMT2A (0.41) PARP1ELANEGRIN1GRIN2AACHE
SCHEMBL25463097 0.71 MAOA (0.52) ACHETDP1
SCHEMBL10455684 0.71 TDP1 (0.46) PARP1ELANEGRIN1GRIN2AACHE
SCHEMBL29145497 0.71 DHODH (0.46) PARP1ELANE
SCHEMBL5234447 0.69 PARP1 (0.41) PARP1ELANEGRIN1GRIN2AACHE
SCHEMBL7811084 0.68 PARP1 (0.46) PARP1ELANEGRIN1GRIN2AACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109641886-A bicyclic BET bromodomain inhibitors and uses thereof 康威基内有限公司 2019-04-16 CN disclosed