SCHEMBL28293716

SCHEMBL28293716

NCc1ccc(-c2ccc(-c3ccc(CN)cc3)o2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.62
TAAR1 Q96RJ0 4/20 0.57
CYP2E1 P05181 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2A6 P11509 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2B6 P20813 1/20 0.48
CYP2C19 P33261 1/20 0.48
LOXL2 Q9Y4K0 3/20 0.46
TOP2A P11388 3/20 0.45
TOP2B Q02880 3/20 0.45
ALDH1A1 P00352 3/20 0.45
HPGD P15428 3/20 0.45
HSD17B10 Q99714 3/20 0.45
ADRB2 P07550 1/20 0.45
TOP1 P11387 1/20 0.45
NQO2 P16083 1/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21381239 0.87 CYP2A6 (0.68) HRH3TAAR1CYP2E1CYP3A4CYP2D6
SCHEMBL13680605 0.85 HRH3 (0.50) HRH3TAAR1CYP2E1CYP3A4CYP2D6
SCHEMBL24670424 0.85 HRH3 (0.50) HRH3TAAR1CYP2E1CYP3A4CYP2D6
SCHEMBL19853627 0.83 NQO2 (0.52) CYP2C9CYP2C19TOP2ATOP2BALDH1A1
SCHEMBL2274647 0.78 HRH3 (1.00) HRH3TAAR1CYP2A6LOXL2ADRB2
SCHEMBL5452549 0.78 HDAC3 (0.56) ALDH1A1HPGDHSD17B10KDM4ENPC1
SCHEMBL15828 0.74 HRH3 (0.79) HRH3TAAR1LOXL2ADRB2ABAT
SCHEMBL112138 0.73 TAAR1 (1.00) HRH3TAAR1CYP2A6LOXL2ADRB2
SCHEMBL34464672 0.72 CA12 (0.57) HRH3TAAR1CYP2A6LOXL2ALDH1A1
SCHEMBL4338939 0.71 CALM1 (0.55) CYP2E1CYP3A4CYP2D6CYP2A6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109705012-A A kind of preparation method of 2,5- diaryl five-ring heterocycles aromatic hydrocarbons 西北师范大学 2019-05-03 CN disclosed