SCHEMBL28294252

SCHEMBL28294252

CNC(=O)c1ccc(C(=O)ON)cn1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.56
KDM4E B2RXH2 3/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
ALDH1A1 P00352 4/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
AHR P35869 1/20 0.43
NNMT P40261 1/20 0.42
BAZ2B Q9UIF8 1/20 0.42
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 1/20 0.41
PIP5K1C O60331 1/20 0.41
PIK3CA P42336 1/20 0.41
PI4KA P42356 1/20 0.41
PI4KB Q9UBF8 1/20 0.41
P4HTM Q9NXG6 6/20 0.41
P4HA1 P13674 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL600512 0.87 MAPK1 (0.74) MAPK1KDM4EL3MBTL1ALDH1A1NPC1
SCHEMBL2219738 0.83 NNMT (0.61) MAPK1KDM4EL3MBTL1ALDH1A1NPC1
SCHEMBL13184552 0.83 BAZ2B (0.57) MAPK1KDM4EL3MBTL1ALDH1A1NPC1
SCHEMBL2113530 0.80 P4HTM (0.66) MAPK1KDM4EL3MBTL1ALDH1A1NPC1
SCHEMBL29967093 0.80 P4HTM (0.66) MAPK1KDM4EL3MBTL1ALDH1A1NPC1
SCHEMBL599587 0.78 P4HTM (0.63) MAPK1KDM4EL3MBTL1ALDH1A1NPC1
SCHEMBL13754096 0.77 GRM5 (0.51) MAPK1KDM4EL3MBTL1ALDH1A1NPC1
SCHEMBL31314624 0.77 MAPK1 (0.74) MAPK1KDM4EL3MBTL1ALDH1A1NPC1
SCHEMBL18231649 0.77 ALDH1A1 (0.47) MAPK1KDM4EL3MBTL1ALDH1A1NPC1
SCHEMBL28650145 0.77 MAPK1 (0.74) MAPK1KDM4EL3MBTL1ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed