SCHEMBL28294492

SCHEMBL28294492

NS(=O)(=O)c1ccc(-n2nc(C(=O)O)cc2-c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.77

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.77
PTGS2 P35354 14/20 0.73
CYP2C9 P11712 1/20 0.73
PTGS1 P23219 6/20 0.71
PDPK1 O15530 4/20 0.71
EPHX2 P34913 2/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5698710 0.87 PTGS2 (0.76) CHRNA7PTGS2PTGS1
SCHEMBL27485652 0.86 PTGS2 (0.65) CHRNA7PTGS2PTGS1
SCHEMBL5236666 0.86 RPA1 (0.72) PTGS2PTGS1EPHX2
SCHEMBL5430032 0.85 CA9 (0.74) CHRNA7PTGS2CYP2C9PTGS1PDPK1
SCHEMBL27485627 0.85 PTGS2 (0.69) CHRNA7PTGS2PTGS1
SCHEMBL3873219 0.85 CHRNA7 (0.80) CHRNA7PTGS2
SCHEMBL3096416 0.84 PTGS2 (1.00) PTGS2CYP2C9PTGS1PDPK1
SCHEMBL8121963 0.83 PTGS2 (0.80) CHRNA7PTGS2CYP2C9PTGS1PDPK1
SCHEMBL5858004 0.83 PDPK1 (1.00) PTGS2CYP2C9PTGS1PDPK1
SCHEMBL16876818 0.83 MEN1 (0.60) CHRNA7PTGS2CYP2C9PTGS1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109748872-A The design and synthesis of the morpholine derivative antitumoral compounds of one kind skeleton containing diaryl pyrazole 南京大学 2019-05-14 CN disclosed