SCHEMBL28294761

SCHEMBL28294761

C1=CN(C2CC2)Cc2ccccc21

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.37
KCNH2 Q12809 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
HDAC3 O15379 1/20 0.35
HSD17B3 P37058 1/20 0.32
SRD5A1 P18405 1/20 0.32
DPP4 P27487 1/20 0.31
FAP Q12884 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP9 Q86TI2 1/20 0.31
DPP7 Q9UHL4 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30364155 0.92 MAPK1 (0.35) PARP1KCNH2HRH3HDAC3DPP4
SCHEMBL19691139 0.92 MAPK1 (0.35) PARP1KCNH2HRH3HDAC3DPP4
SCHEMBL30399174 0.88 HTR2C (0.42) PARP1HDAC3
SCHEMBL29874963 0.82 DRD2 (0.35) KCNH2
SCHEMBL28807401 0.80 PARP1 (0.39) PARP1
SCHEMBL29875020 0.76 CYP3A4 (0.32)
SCHEMBL3069885 0.73 HDAC3 (0.43) PARP1KCNH2HDAC3HSD17B3CA1
SCHEMBL7237449 0.72 HTR2C (0.34) PARP1HDAC3
SCHEMBL5360614 0.71 PARP1 (0.37) PARP1HDAC3
SCHEMBL5819959 0.70 PRCP (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105130966-B Alkynyl compounds and its application method and purposes 广东东阳光药业有限公司 2019-05-24 CN disclosed