SCHEMBL5819959

SCHEMBL5819959

C1=CN(C2NCCc3ccccc32)Cc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PRCP P42785 8/20 0.43
GAA P10253 2/20 0.42
SLC22A1 O15245 1/20 0.39
RECQL P46063 1/20 0.39
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
GID4 Q8IVV7 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
MAPT P10636 1/20 0.35
OPRM1 P35372 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15473972 0.77 PRCP (0.43) PRCPGAASLC22A1RECQLTSHR
SCHEMBL5360614 0.75 PARP1 (0.37) HTR2A
SCHEMBL4276041 0.72 PRCP (0.44) PRCPGAASLC22A1RECQLTSHR
SCHEMBL27814188 0.71 CYP1A2 (0.39) GAAHTR2A
SCHEMBL18093730 0.70 CYP2D6 (0.33) TSHRKDM4EALDH1A1MAPT
SCHEMBL30399174 0.70 HTR2C (0.42) HTR2AHTR2CHTR2B
SCHEMBL28294761 0.70 PARP1 (0.37)
SCHEMBL30345136 0.69 PRCP (0.41) PRCPGAASLC22A1RECQLTSHR
SCHEMBL5571017 0.68 PRCP (0.51) PRCPGAASLC22A1RECQLTSHR
SCHEMBL27898029 0.68 HTR2C (0.39) HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1723134-A2 TETRAHYDROISOQUINOLINYL DERIVATIVES OF QUINAZOLINE AND ISOQUINOLINE Pfizer Products Incorporated (US) 2006-11-22 EP disclosed
WO-2005082883-A2 TETRAHYDROISOQUINOLINYL DERIVATIVES OF QUINAZOLINE AND ISOQUINOLINE PFIZER PRODUCTS INC. (US) 2005-09-09 WO disclosed