SCHEMBL28295038

SCHEMBL28295038

N#Cc1cc(-c2[c]cccn2)ccc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.41
FLT3 P36888 2/20 0.41
CYP11B2 P19099 4/20 0.39
CNR2 P34972 1/20 0.39
PDE10A Q9Y233 1/20 0.36
PGR P06401 2/20 0.36
LRRK2 Q5S007 1/20 0.36
CYP11B1 P15538 3/20 0.36
MAOB P27338 1/20 0.36
PIK3CD O00329 1/20 0.36
ABL1 P00519 1/20 0.36
EGFR P00533 1/20 0.36
HCK P08631 1/20 0.36
SRC P12931 1/20 0.36
KDR P35968 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
MTOR P42345 1/20 0.36
PIK3CG P48736 1/20 0.36
EPHB4 P54760 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5541420 0.81 CYP17A1 (0.41) CYP11B2CYP11B1MAOB
SCHEMBL1514336 0.78 CLK4 (0.51) GRM4FLT3CYP11B2CNR2PDE10A
SCHEMBL5542548 0.77 NISCH (0.42) GRM4CYP11B2KDRPIK3CAEPHB4
SCHEMBL28413182 0.77 GRIN2B (0.40) GRM4FLT3LRRK2KDR
SCHEMBL28138779 0.76 GRIN2B (0.39)
SCHEMBL5290073 0.74 CYP11B2 (0.43) CYP11B2
SCHEMBL1965066 0.74 CLK4 (0.60) MAOB
SCHEMBL5330919 0.74 CNR2 (0.44) GRM4FLT3CYP11B2CNR2PGR
SCHEMBL2668166 0.74 CNR2 (0.47) GRM4FLT3CYP11B2CNR2PDE10A
SCHEMBL2656644 0.74 GRM4 (0.50) GRM4FLT3CYP11B2CNR2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104837832-B GDF-8 inhibitors 里格尔药品股份有限公司 2019-04-26 CN claimed
CN-106536507-B 2, 3-disubstituted pyridine compounds as TGF- β inhibitors and methods of use thereof 里格尔药品股份有限公司 2020-04-07 CN disclosed
CN-104837832-B GDF-8 inhibitors 里格尔药品股份有限公司 2019-04-26 CN disclosed