SCHEMBL5290073

SCHEMBL5290073

N#Cc1ccc(-c2[c]cccn2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.43
CLK4 Q9HAZ1 1/20 0.40
HSD11B1 P28845 1/20 0.39
MMP3 P08254 1/20 0.38
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
NPY5R Q15761 1/20 0.37
SLC6A7 Q99884 1/20 0.37
CYP19A1 P11511 3/20 0.37
EGLN2 Q96KS0 2/20 0.36
TDO2 P48775 1/20 0.36
SLC11A2 P49281 1/20 0.36
SLC22A12 Q96S37 1/20 0.36
NOTUM Q6P988 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1965066 0.81 CLK4 (0.60) CLK4EGLN2NOTUM
SCHEMBL1202054 0.77 NOTUM (0.37) NPY5RNOTUM
SCHEMBL5539865 0.76 NISCH (0.37) SLC6A7
SCHEMBL1973038 0.76 MAPK14 (0.36) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL435455 0.76 CYP1A2 (0.38) CYP19A1NOTUM
SCHEMBL1980545 0.76 ALDH1A1 (0.38) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL2397171 0.75 MAPT (0.42) CYP11B2NPY5RCYP19A1NOTUMKIF11
SCHEMBL28295038 0.74 GRM4 (0.41) CYP11B2
SCHEMBL3996884 0.74 CYP11B2 (0.41) CYP11B2CLK4NPY5RCYP19A1
SCHEMBL1741768 0.72 CLK4 (0.62) CYP11B2CLK4HSD11B1MMP3CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103864677-B Thioacetic acid salt compound, compoistion and method of use ARDEA BIOSCIENCES, INC. (US) 2016-05-18 CN disclosed
CN-103864677-A THIOACETATE COMPOUNDS, COMPOSITIONS AND METHODS OF USE ARDEA BIOSCIENCES INC 2014-06-18 CN disclosed
CN-103068801-B Thioacetate compounds, compositions, and methods of use ARDEA BIOSCIENCES INC 2014-05-14 CN disclosed
EP-1861411-A2 NOVEL COMPOUNDS DERIVED FROM 5-THIOXYLOSE AND THERAPEUTIC USE THEREOF LABORATOIRES FOURNIER S.A. (FR) 2007-12-05 EP disclosed
WO-2006100413-A9 NOVEL COMPOUNDS DERIVED FROM 5-THIOXYLOSE AND THERAPEUTIC USE THEREOF FOURNIER LAB SA (FR) 2007-10-18 WO disclosed
WO-2006100413-A2 NOVEL COMPOUNDS DERIVED FROM 5-THIOXYLOSE AND THERAPEUTIC USE THEREOF LABORATOIRES FOURNIER S.A. (FR) 2006-09-28 WO disclosed