SCHEMBL28295466

SCHEMBL28295466

CCC1CNc2ccc(N)cc2C(c2ccccc2F)=N1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 4/20 0.49
CHRM1 P11229 4/20 0.40
CHRM5 P08912 1/20 0.40
TRPV1 Q8NER1 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28297189 0.88 CCKBR (0.60) CCKBRCHRM1CHRM5
SCHEMBL28297206 0.81 CCKBR (0.48) CCKBRCHRM1TRPV1
Bromide SCHEMBL9526214 0.76 CCKBR (0.59) CCKBRCHRM1
Bromide SCHEMBL9526221 0.76 CCKBR (0.59) CCKBRCHRM1
SCHEMBL21272067 0.76 CHRM1 (0.56) CHRM1CHRM5TRPV1
SCHEMBL28295476 0.72 CHRM1 (0.61) CHRM1CHRM5TRPV1
SCHEMBL28297200 0.72 CHRM1 (0.61) CHRM1CHRM5TRPV1
SCHEMBL28297188 0.72 CHRM1 (0.49) CCKBRCHRM1
SCHEMBL11265240 0.71 GABRA1 (0.52) CCKBRCHRM1CHRM5TRPV1
SCHEMBL28297201 0.71 CHRM1 (0.46) CCKBRCHRM1CHRM5TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109906220-A For treating the 1,3- dihydro -1,4- benzodiazepine * -2- thione compounds of CNS related disease 豪夫迈·罗氏有限公司 2019-06-18 CN claimed
CN-109906220-A For treating the 1,3- dihydro -1,4- benzodiazepine * -2- thione compounds of CNS related disease 豪夫迈·罗氏有限公司 2019-06-18 CN disclosed