Pyrazole

Pyrazole

SCHEMBL28295801

Fc1ccncc1F.c1cn[nH]c1

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.37
NUDT1 P36639 2/20 0.37
CDC7 O00311 1/20 0.33
ROCK2 O75116 1/20 0.33
MAP4K4 O95819 1/20 0.33
PRKACA P17612 1/20 0.33
CDK2 P24941 1/20 0.33
GSK3B P49841 1/20 0.33
HIPK2 Q9H2X6 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
RPS6KA3 P51812 1/20 0.31
CYP1A2 P05177 1/20 0.31
METAP2 P50579 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29518741 0.78
SCHEMBL3717170 0.78
Pyrazole SCHEMBL28114392 0.74 SCN4A (0.37)
Isoquinoline SCHEMBL1133594 0.73 MAPT (0.38) CYP1A2
Imidazole SCHEMBL28295853 0.72 ALDH1A1 (0.54) LOXL2NUDT1
Pyrazole SCHEMBL16874402 0.72
Pyrazole SCHEMBL30626480 0.71
Pyrazole SCHEMBL30854861 0.71
Pyrazole SCHEMBL5664483 0.71
Pyrazole SCHEMBL1384 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106232600-B Indolin-2-one and 1,3- dihydro-pyrrole simultaneously [3,2-c] pyridin-2-ones derivative 豪夫迈·罗氏有限公司 2019-05-14 CN disclosed