SCHEMBL28296044

SCHEMBL28296044

CC(C)(C)OC(=O)c1c(F)c[c]cc1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM6 O15303 1/20 0.35
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MAPT P10636 2/20 0.33
TP53 P04637 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
NR1H2 P55055 2/20 0.32
NR1H3 Q13133 2/20 0.32
RXRA P19793 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL679324 0.78 GAA (0.45) GRM6CYP2C9CYP2C19NPSR1CA12
SCHEMBL25304437 0.77 CYP2C9 (0.37) GRM6CYP2C9CYP2C19NPSR1CA12
SCHEMBL14289250 0.77 CYP2C9 (0.47) GRM6CYP2C9CYP2C19NPSR1CA12
SCHEMBL15359768 0.76 GRM6 (0.40) GRM6CYP2C9CYP2C19NPSR1MAPT
SCHEMBL643173 0.76 AAK1 (0.39) GRM6CYP2C9CYP2C19NPSR1MAPT
SCHEMBL20741090 0.75 NR3C2 (0.41) CYP2C9CYP2C19NPSR1GABRA1GABRG2
SCHEMBL27768243 0.75 NR3C2 (0.34) MAPTCA12CA1CA2CA9
SCHEMBL522898 0.74 TSHR (0.37) GRM6CYP2C9CYP2C19NPSR1CA12
SCHEMBL5774469 0.74 AKR1C3 (0.42) GRM6CYP2C9CYP2C19NPSR1CA1
SCHEMBL20741075 0.74 LMNA (0.42) GRM6CYP2C9CYP2C19NPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715633-A Dopamine-B-hydroxylase inhibitors 巴尔-波特拉及康邦亚股份有限公司 2019-05-03 CN disclosed