SCHEMBL28296065

SCHEMBL28296065

CCC(=O)Cc1ncc(C(=O)OC)[nH]1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.56
BAZ2B Q9UIF8 1/20 0.39
BAZ2A Q9UIF9 1/20 0.39
ALDH1A1 P00352 3/20 0.36
MAPK1 P28482 2/20 0.36
CYP1A2 P05177 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
GAA P10253 2/20 0.35
KDM4E B2RXH2 1/20 0.35
GLA P06280 1/20 0.35
XDH P47989 1/20 0.35
ALPL P05186 1/20 0.34
ABL1 P00519 8/20 0.33
SRC P12931 8/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28296067 0.84 MMP2 (0.58) MMP2BAZ2BBAZ2AALDH1A1MAPK1
SCHEMBL7424608 0.83 MMP2 (0.61) MMP2BAZ2BBAZ2AALDH1A1MAPK1
SCHEMBL8653203 0.81 MMP2 (0.67) MMP2BAZ2BBAZ2AALDH1A1MAPK1
SCHEMBL4605593 0.79 MMP2 (0.60) MMP2ALDH1A1MAPK1CYP1A2NPC1
SCHEMBL20630811 0.79 MMP2 (0.60) MMP2BAZ2BBAZ2AALDH1A1MAPK1
SCHEMBL31373939 0.78 MMP2 (0.58) MMP2BAZ2BBAZ2AALDH1A1MAPK1
SCHEMBL14744177 0.78 MMP2 (0.67) MMP2BAZ2BBAZ2AALDH1A1MAPK1
Hydrochloric Acid SCHEMBL14744176 0.76 MMP2 (0.65) MMP2ALDH1A1MAPK1CYP1A2GAA
SCHEMBL9605532 0.75 MMP2 (0.56) MMP2BAZ2BBAZ2AALDH1A1MAPK1
SCHEMBL28193948 0.73 KDM6B (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107531714-B Imidazopyrazines ketone as PDE1 inhibitor H.隆德贝克有限公司 2019-07-19 CN disclosed
CN-109803658-A Combined therapy comprising the Imidazopyrazines ketone for treating mental disease and/or cognitive disorder H.隆德贝克有限公司 2019-05-24 CN disclosed
CN-109803653-A Combined therapy including giving Imidazopyrazines ketone H.隆德贝克有限公司 2019-05-24 CN disclosed
CN-107531714-A Imidazopyrazines ketone as PDE1 inhibitor H.隆德贝克有限公司 2018-01-02 CN disclosed