SCHEMBL28296308

SCHEMBL28296308

N=C(Nc1ccccc1)c1ccc(C(F)(F)F)cc1/C=C/c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.42
MAPT P10636 4/20 0.42
KMT2A Q03164 4/20 0.42
RAB9A P51151 3/20 0.42
HTT P42858 1/20 0.42
LMNA P02545 2/20 0.40
PAX8 Q06710 1/20 0.40
HSP90AA1 P07900 1/20 0.40
PKM P14618 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
NPC1 O15118 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAOB P27338 3/20 0.39
KCNK3 O14649 1/20 0.39
GPR27 Q9NS67 4/20 0.38
AVPR2 P30518 3/20 0.38
GRIK1 P39086 1/20 0.38
CYP1A1 P04798 1/20 0.38
CYP1B1 Q16678 1/20 0.38
TRPA1 O75762 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28294692 0.91 MEN1 (0.39) MEN1MAPTKMT2ARAB9AHTT
SCHEMBL28296314 0.80 MAOB (0.44) MEN1MAPTKMT2ARAB9ALMNA
SCHEMBL28571714 0.77 GPR27 (0.55) MEN1MAPTKMT2ARAB9AHTT
SCHEMBL28576258 0.74 JAK2 (0.52) MEN1MAPTKMT2ARAB9AHTT
SCHEMBL28417758 0.73 GRIN1 (0.43) MEN1KMT2AMAOBCYP1A1CYP1B1
SCHEMBL28417757 0.73 GRIN1 (0.43) MEN1KMT2AMAOBCYP1A1CYP1B1
SCHEMBL28294691 0.73 GRIN1 (0.43) MEN1KMT2AMAOBCYP1A1CYP1B1
SCHEMBL28415675 0.70 RAB9A (0.57) MEN1MAPTKMT2ARAB9AHTT
SCHEMBL16400445 0.69 MAOB (0.46) MAPTRAB9AMAOBCYP1A1CYP1B1
SCHEMBL16400448 0.69 MAOB (0.46) MAPTRAB9AMAOBCYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109796372-A A method of preparing polysubstituted alkenyl amidine 中国科学院化学研究所 2019-05-24 CN disclosed