SCHEMBL28296323

SCHEMBL28296323

NC(=Nc1ccccc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.66
KMT2A Q03164 1/20 0.66
CYP2D6 P10635 1/20 0.61
HIF1A Q16665 1/20 0.61
GRIN2B Q13224 5/20 0.59
HTR3E A5X5Y0 3/20 0.56
HTR3B O95264 3/20 0.56
HTR3A P46098 3/20 0.56
HTR3D Q70Z44 3/20 0.56
HTR3C Q8WXA8 3/20 0.56
PLAU P00749 2/20 0.56
NOS1 P29475 6/20 0.47
NOS3 P29474 4/20 0.47
PRSS1 P07477 1/20 0.47
ACR P10323 1/20 0.47
SLC22A2 O15244 1/20 0.45
SLC22A1 O15245 1/20 0.45
SLC22A3 O75751 1/20 0.45
ALDH1A1 P00352 3/20 0.45
LMNA P02545 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8398110 0.93 MEN1 (0.66) MEN1KMT2ACYP2D6HIF1AGRIN2B
SCHEMBL28216626 0.81 KMT2A (0.59) MEN1KMT2ACYP2D6HIF1AHTR3E
SCHEMBL24662980 0.80 KMT2A (1.00) MEN1KMT2ACYP2D6HIF1AGRIN2B
SCHEMBL139363 0.80 KMT2A (1.00) MEN1KMT2ACYP2D6HIF1AGRIN2B
SCHEMBL24136574 0.80 KMT2A (1.00) MEN1KMT2ACYP2D6HIF1AGRIN2B
SCHEMBL4863419 0.79 NOS1 (0.56) MEN1KMT2ACYP2D6HIF1AGRIN2B
SCHEMBL13819189 0.79 HTR3E (0.47) GRIN2BHTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL28549744 0.78 KMT2A (0.95) MEN1KMT2ACYP2D6HIF1AGRIN2B
Hydrochloric Acid SCHEMBL9773794 0.78 KMT2A (0.95) MEN1KMT2ACYP2D6HIF1AGRIN2B
SCHEMBL5594042 0.77 AKR1C3 (0.50) KMT2AGRIN2BHTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109796372-A A method of preparing polysubstituted alkenyl amidine 中国科学院化学研究所 2019-05-24 CN disclosed