SCHEMBL28296698

SCHEMBL28296698

Oc1ccccc1-c1cccc2cc(F)ccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.45
CYP2A6 P11509 1/20 0.45
HSD17B1 P14061 5/20 0.45
HSD17B2 P37059 5/20 0.45
CASR P41180 3/20 0.42
PLAU P00749 1/20 0.42
LMNA P02545 2/20 0.40
TP53 P04637 2/20 0.40
MAPT P10636 2/20 0.40
ALOX15 P16050 2/20 0.40
MAPK1 P28482 2/20 0.40
ALOX12 P18054 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ESR1 P03372 3/20 0.40
ESR2 Q92731 3/20 0.40
TLR8 Q9NR97 1/20 0.40
MEN1 O00255 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18530961 0.87 CYP1A2 (0.52) CYP1A2CYP2A6HSD17B1HSD17B2MAPK1
SCHEMBL29549050 0.85 CYP1A2 (0.52) CYP1A2CYP2A6MAPK1KDM4ETSHR
SCHEMBL2529937 0.83 HSD17B1 (0.59) CYP1A2CYP2A6HSD17B1HSD17B2PLAU
SCHEMBL31556780 0.83 HSD17B1 (0.59) CYP1A2CYP2A6HSD17B1HSD17B2PLAU
SCHEMBL27607735 0.79 PLAU (0.70) CYP1A2HSD17B1HSD17B2PLAULMNA
SCHEMBL18529228 0.79 CYP2A6 (0.45) CYP1A2CYP2A6HSD17B1HSD17B2PLAU
SCHEMBL29291191 0.79 CYP2A6 (0.45) CYP1A2CYP2A6HSD17B1HSD17B2CASR
SCHEMBL29291203 0.79 CYP1A2 (0.53) CYP1A2CYP2A6HSD17B1HSD17B2PLAU
SCHEMBL30214159 0.78 CYP1A2 (0.65) CYP1A2CYP2A6HSD17B1HSD17B2TP53
SCHEMBL217637 0.78 CYP1A2 (0.65) CYP1A2CYP2A6HSD17B1HSD17B2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843856-A KRAS G12C inhibitor 米拉蒂治疗股份有限公司 2019-06-04 CN disclosed
CN-109715632-A Macrocyclic indole derivatives 拜尔公开股份有限公司 2019-05-03 CN disclosed