SCHEMBL28296838

SCHEMBL28296838

Fc1cc(F)cc([C@H]2CCNC2)c1.NC=S

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.43
MPO P05164 1/20 0.38
HRH4 Q9H3N8 1/20 0.36
PDE4B Q07343 1/20 0.35
HTR2C P28335 1/20 0.35
CYP2D6 P10635 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28298499 1.00 HTR3A (0.43) HTR3AMPOHRH4PDE4BHTR2C
SCHEMBL28873365 1.00 HTR3A (0.43) HTR3AMPOHRH4PDE4BHTR2C
SCHEMBL21527890 0.91 HTR3A (0.50) HTR3AMPOPDE4BCYP2D6SLC6A2
SCHEMBL1822208 0.91 HTR3A (0.50) HTR3AMPOPDE4BCYP2D6SLC6A2
SCHEMBL21527834 0.91 HTR3A (0.50) HTR3AMPOPDE4BCYP2D6SLC6A2
SCHEMBL28296843 0.83 HTR3A (0.38) HTR3AMPOHTR2CSLC6A2SLC6A4
SCHEMBL28298501 0.83 HTR3A (0.56) HTR3AMPOHTR2C
SCHEMBL24127329 0.82 DRD2 (0.47) HTR2CCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL28873499 0.80 HCAR2 (0.38) HTR3AMPOHTR2C
SCHEMBL1823726 0.79 HTR3A (0.56) HTR3ACYP2D6SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715155-A blood brain barrier-penetrating agent dopamine- β -hydroxylase inhibitors 巴尔-波特拉及康邦亚股份有限公司 2019-05-03 CN disclosed