SCHEMBL28296983

SCHEMBL28296983

COC(=O)CC(c1ccc(F)cc1F)C(C)C(=O)OC#N

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.35
HTT P42858 1/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
PKM P14618 1/20 0.33
POLB P06746 1/20 0.33
LGMN Q99538 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19972301 0.81 ALDH1A1 (0.36) ALDH1A1MAPTHTTPSEN1PSEN2
SCHEMBL12525150 0.72 MAPT (0.46) ALDH1A1MAPTHTTCES2CES1
SCHEMBL19972227 0.70 KMT2A (0.38) ALDH1A1MAPT
SCHEMBL756201 0.69 HTT (0.32) ALDH1A1MAPTHTT
SCHEMBL9997229 0.69 CES2 (0.42) ALDH1A1MAPTPSEN1PSEN2APH1B
SCHEMBL31117167 0.68 CES2 (0.46) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL31560789 0.68 CES2 (0.46) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL19985861 0.67 KMT2A (0.38) ALDH1A1MAPT
SCHEMBL4533837 0.67 CES2 (0.45) ALDH1A1MAPTHTTPSEN1PSEN2
SCHEMBL15499253 0.67 ALDH1A1 (0.36) ALDH1A1MAPTHTTPSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715614-A The 6 yuan of cyclammonium or lactams replaced with urea and phenyl 格吕伦塔尔有限公司 2019-05-03 CN disclosed