SCHEMBL28297464

SCHEMBL28297464

Cc1c(CCCCCl)cccc1C(N)=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
PARP1 P09874 6/20 0.37
CYP3A4 P08684 2/20 0.37
NR1I2 O75469 1/20 0.37
LMNA P02545 1/20 0.37
CHRM2 P08172 1/20 0.37
ADRA2A P08913 1/20 0.37
MAPT P10636 1/20 0.37
OPRK1 P41145 1/20 0.37
HTR2B P41595 1/20 0.37
SLC6A3 Q01959 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
CD38 P28907 3/20 0.37
SIRT2 Q8IXJ6 2/20 0.37
MRGPRX4 Q96LA9 1/20 0.36
AURKA O14965 1/20 0.36
RPS6KB1 P23443 1/20 0.36
SLC16A3 O15427 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28298922 0.95 MEN1 (0.38) MEN1KMT2AKDM4EPARP1CYP3A4
SCHEMBL28232396 0.89 KDM4E (0.40) MEN1KMT2AKDM4EPARP1CYP3A4
SCHEMBL6013407 0.86 BID (0.48) MEN1KMT2AKDM4ECYP3A4NR1I2
SCHEMBL7517986 0.84 BID (0.50) MEN1KMT2AKDM4ECYP3A4NR1I2
SCHEMBL6013409 0.84 BID (0.50) MEN1KMT2AKDM4ECYP3A4NR1I2
SCHEMBL486383 0.84 MEN1 (0.45) MEN1KMT2AKDM4EPARP1CYP3A4
SCHEMBL30514834 0.84 PARP1 (0.38) MEN1KMT2AKDM4EPARP1CYP3A4
SCHEMBL28182515 0.84 PARP1 (0.38) MEN1KMT2AKDM4EPARP1CYP3A4
SCHEMBL29009406 0.83 MAPT (0.42) MEN1KMT2AKDM4EPARP1CYP3A4
Hydrochloric Acid SCHEMBL7557316 0.83 BID (0.49) MEN1KMT2AKDM4ECYP3A4NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109863146-A Aryl-linking compound as immunomodulator 百时美施贵宝公司 2019-06-07 CN disclosed