SCHEMBL28297598

SCHEMBL28297598

COC(=O)Nc1ccc(Br)c(N)c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 3/20 0.45
MAPT P10636 2/20 0.44
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
HPGD P15428 1/20 0.44
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
TDP1 Q9NUW8 1/20 0.42
FAAH O00519 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPK1 P28482 1/20 0.41
PKM P14618 2/20 0.41
GAA P10253 1/20 0.41
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29780101 1.00 SMN1; SMN2 (0.50) SMN1; SMN2ALDH1A1MAPTRAB9ANPC1
SCHEMBL28599978 0.84 CA12 (0.47) SMN1; SMN2ALDH1A1RAB9ANPC1GAA
SCHEMBL26617403 0.84 KDM4E (0.57) SMN1; SMN2ALDH1A1MAPTRAB9ANPC1
SCHEMBL29780064 0.84 CA12 (0.47) SMN1; SMN2ALDH1A1RAB9ANPC1GAA
SCHEMBL4606482 0.82 TDP1 (0.55) SMN1; SMN2ALDH1A1MAPTRAB9ANPC1
SCHEMBL10782684 0.81 SMN1; SMN2 (0.52) SMN1; SMN2ALDH1A1MAPTHPGDKMT2A
SCHEMBL31314406 0.81 SMN1; SMN2 (0.52) SMN1; SMN2ALDH1A1MAPTHPGDKMT2A
SCHEMBL21262587 0.81 SMN1; SMN2 (0.52) SMN1; SMN2ALDH1A1MAPTRAB9ANPC1
SCHEMBL29965600 0.81 SMN1; SMN2 (0.52) SMN1; SMN2ALDH1A1MAPTRAB9ANPC1
SCHEMBL3928807 0.81 ALDH1A1 (0.67) SMN1; SMN2ALDH1A1MAPTRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108430471-B Factor XIa inhibitors 默沙东公司 2021-07-09 CN disclosed
CN-109721613-A Macro-cyclic amide compound and its pharmaceutical composition and purposes containing quaternary ammonium ion 四川科伦博泰生物医药股份有限公司 2019-05-07 CN disclosed