SCHEMBL28297925

SCHEMBL28297925

O=C(O)C1CC(c2ccc(C(F)F)cc2)=NN(c2cccc(F)c2)C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 3/20 0.39
NR3C2 P08235 2/20 0.38
NT5E P21589 1/20 0.37
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
MAOB P27338 2/20 0.36
MAOA P21397 1/20 0.36
CACNA1C Q13936 1/20 0.35
PTGS2 P35354 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
GAA P10253 2/20 0.35
HSP90AA1 P07900 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19642149 0.88 PDE4A (0.39) CACNA1HNR3C2NT5EKDM4EALDH1A1
SCHEMBL30187402 0.88 PDE4A (0.39) CACNA1HNR3C2NT5EKDM4EALDH1A1
SCHEMBL28299533 0.87 KDM4E (0.41) CACNA1HNR3C2NT5EKDM4EALDH1A1
SCHEMBL28299380 0.84 MEN1 (0.49) CACNA1HNR3C2NT5EKDM4EALDH1A1
SCHEMBL28873447 0.84 KDM4E (0.51) CACNA1HNR3C2KDM4EALDH1A1PDE4A
SCHEMBL19659889 0.84 PDE4A (0.51) CACNA1HNR3C2KDM4EALDH1A1PDE4A
SCHEMBL28297923 0.82 MEN1 (0.41) CACNA1HNR3C2KDM4EPDE4APDE4B
SCHEMBL28299379 0.78 MAOB (0.41) KDM4EALDH1A1MAOBMAOAPTGS2
SCHEMBL28297928 0.77 NT5E (0.35) CACNA1HNR3C2NT5EKDM4EALDH1A1
SCHEMBL30187450 0.76 KDM4E (0.41) CACNA1HKDM4EALDH1A1PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109863140-A 3- oxo -2,6- diphenyl -2,3- dihydrogen dazin -4- formamide 拜耳医药股份有限公司 2019-06-07 CN disclosed