SCHEMBL28298079

SCHEMBL28298079

O=COCc1cccc(CBr)n1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.40
CCR1 P32246 1/20 0.36
LMNA P02545 1/20 0.36
PGK1 P00558 1/20 0.33
PGK2 P07205 1/20 0.33
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27788777 0.81 KCNH2 (0.36) KCNH2LMNA
SCHEMBL28659624 0.81 KCNH2 (0.40) KCNH2LMNAPGK1PGK2NPSR1
SCHEMBL27600750 0.78 BACE1 (0.39) KCNH2LMNA
SCHEMBL5924102 0.78 SMN1; SMN2 (0.41) KCNH2CCR1
SCHEMBL28119095 0.78 CYP3A4 (0.38) KCNH2LMNA
SCHEMBL28072140 0.78 CCR1 (0.36) KCNH2CCR1LMNA
SCHEMBL245158 0.77 CCR1 (0.55) KCNH2CCR1LMNAPGK1PGK2
SCHEMBL28332129 0.75 KDM1A (0.40) KCNH2
Bromide SCHEMBL1259355 0.75 CCR1 (0.52) KCNH2CCR1LMNAPGK1PGK2
SCHEMBL2082787 0.75 KCNH2 (0.44) KCNH2CCR1LMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843891-A Oxadiazolopyridine derivatives as ghrelin O-acyltransferase (GOAT) inhibitors 勃林格殷格翰国际有限公司 2019-06-04 CN disclosed
CN-104230827-B 1-(aryl methyl) quinazoline-2,4 (1H, 3H)-diketone is as PARP inhibitor and application thereof 南京英派药业有限公司 2016-10-26 CN disclosed