SCHEMBL28298101

SCHEMBL28298101

Nc1ncc2cc(-c3ccccc3Cl)ccc2n1

nearest known ligand 0.69

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LCK P06239 4/20 0.69
JAK3 P52333 2/20 0.69
KDR P35968 1/20 0.69
MAPK14 Q16539 1/20 0.69
BACE1 P56817 1/20 0.64
ADORA1 P30542 4/20 0.49
TRPA1 O75762 1/20 0.49
ABL1 P00519 3/20 0.48
DHFR P00374 3/20 0.48
ADORA2A P29274 3/20 0.46
ALOX5AP P20292 1/20 0.46
FEN1 P39748 1/20 0.46
USP7 Q93009 1/20 0.46
SRC P12931 3/20 0.45
KIT P10721 2/20 0.45
JAK2 O60674 1/20 0.44
JAK1 P23458 1/20 0.44
TYK2 P29597 1/20 0.44
FGFR1 P11362 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5491016 0.84 LCK (0.56) LCKJAK3KDRMAPK14BACE1
SCHEMBL5494572 0.84 LCK (0.56) LCKJAK3KDRMAPK14BACE1
SCHEMBL5491730 0.83 LCK (0.55) LCKJAK3KDRMAPK14BACE1
SCHEMBL5494575 0.82 LCK (1.00) LCKJAK3KDRMAPK14BACE1
SCHEMBL41115 0.81 LCK (0.53) LCKJAK3KDRMAPK14BACE1
SCHEMBL2741576 0.79 LCK (0.65) LCKJAK3KDRMAPK14BACE1
SCHEMBL5494660 0.78 LCK (0.64) LCKJAK3KDRMAPK14ABL1
SCHEMBL41400 0.78 LCK (0.53) LCKJAK3KDRMAPK14ADORA1
SCHEMBL21416857 0.77 LCK (0.49) LCKJAK3KDRMAPK14ABL1
SCHEMBL5492624 0.77 LCK (0.59) LCKJAK3KDRMAPK14BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843858-A Certain chemical entities, composition and method 润新生物公司 2019-06-04 CN disclosed