SCHEMBL28301259

SCHEMBL28301259

NC(=O)c1cnncc1CCl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.36
NNMT P40261 5/20 0.33
SIRT3 Q9NTG7 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
SIRT6 Q8N6T7 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30
PLK4 O00444 1/20 0.30
CHEK1 O14757 1/20 0.30
AURKA O14965 1/20 0.30
DAPK3 O43293 1/20 0.30
MAP4K4 O95819 1/20 0.30
CSF1R P07333 1/20 0.30
RET P07949 1/20 0.30
FGFR1 P11362 1/20 0.30
PDGFRA P16234 1/20 0.30
LTK P29376 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15095256 0.77 SIRT3 (0.43) TSHRNNMTSIRT3TDP1SIRT6
SCHEMBL1004137 0.68 KDM4E (0.50) TSHRTDP1KDM4EALDH1A1MAPT
SCHEMBL29804459 0.67 SIRT3 (0.55) TSHRNNMTSIRT3TDP1KDM4E
SCHEMBL6075761 0.64 KDM4E (0.41) TSHRKDM4EALDH1A1MAPTHPGD
SCHEMBL27377658 0.64 NNMT (0.36) TSHRNNMTSIRT3TDP1KDM4E
Methane SCHEMBL27687947 0.61 ASPH (0.41) SIRT3TDP1MAP4K4CDK5
SCHEMBL25255537 0.61 PLAU (0.37) SIRT6KDM4EALDH1A1CHEK1AURKA
SCHEMBL17442725 0.60 KDM4C (0.53) TDP1KDM4EALDH1A1MAPT
SCHEMBL9002466 0.60 SIRT3 (0.61) SIRT3TDP1SIRT6KDM4EALDH1A1
SCHEMBL5204576 0.60 TSHR (0.44) TSHRNNMTSIRT3TDP1SIRT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109863139-A Muscarinic acetylcholine receptor M4Positive allosteric modulators of 范德比尔特大学 2019-06-07 CN disclosed