SCHEMBL28307666

SCHEMBL28307666

Cc1c(OB(O)O)cccc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 1/20 0.40
TAS2R14 Q9NYV8 1/20 0.38
HSD11B1 P28845 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PPARG P37231 2/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
SCN8A Q9UQD0 1/20 0.35
MGLL Q99685 1/20 0.34
AR P10275 2/20 0.34
NOTUM Q6P988 1/20 0.34
CTSS P25774 1/20 0.34
DHODH Q02127 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30198749 0.83 PPARG (0.42) HSD11B1MRGPRX4ADRA2AADRA2BADRA2C
SCHEMBL1070284 0.83 PPARG (0.42) HSD11B1MRGPRX4ADRA2AADRA2BADRA2C
SCHEMBL28978849 0.81 PPARG (0.41) HSD11B1MRGPRX4ADRA2AADRA2BADRA2C
SCHEMBL28991513 0.80 MRGPRX4 (0.36) HSD11B1MRGPRX4MEN1KMT2APPARG
SCHEMBL6291525 0.80 MRGPRX4 (0.36) HSD11B1MRGPRX4ADRA2AADRA2BADRA2C
SCHEMBL29515498 0.80 MRGPRX4 (0.36) HSD11B1MRGPRX4ADRA2AADRA2BADRA2C
SCHEMBL28941521 0.80 SCN8A (0.41) TAS2R14HSD11B1MEN1KMT2ASCN8A
SCHEMBL30527011 0.80 IDO1 (0.36) HSD11B1MRGPRX4PPARGRXRARXRB
SCHEMBL7591797 0.80 IDO1 (0.36) HSD11B1MRGPRX4PPARGRXRARXRB
SCHEMBL7593287 0.79 MRGPRX4 (0.35) HSD11B1MRGPRX4ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110062761-A Substituted 1H-imidazo [4,5-b ] pyridin-2 (3H) -ones and their use as GLUN2B receptor modulators 詹森药业有限公司 2019-07-26 CN disclosed