SCHEMBL28313382

SCHEMBL28313382

FC(F)(F)c1cnc(Cl)nc1-c1cccc2cc[nH]c12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.44
CDK1 P06493 1/20 0.39
KDR P35968 1/20 0.39
TRPV1 Q8NER1 2/20 0.38
KDM4E B2RXH2 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PTPN11 Q06124 1/20 0.37
CCNT1 O60563 3/20 0.36
CCNK O75909 3/20 0.36
CDK9 P50750 3/20 0.36
CDK12 Q9NYV4 3/20 0.36
CCNE1 P24864 2/20 0.36
CDK2 P24941 2/20 0.36
REN P00797 2/20 0.34
NR1H2 P55055 1/20 0.34
NR3C1 P04150 3/20 0.33
DYRK1A Q13627 1/20 0.33
RPS6KA5 O75582 1/20 0.33
TNF P01375 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30456841 0.74 CCNT1 (0.59) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL24900464 0.73 CCNT1 (0.48) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL30957488 0.73 CCNT1 (0.48) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL30221492 0.73 CCNT1 (0.57) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL17696390 0.73 CCNT1 (0.57) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL29492558 0.73 CCNT1 (0.57) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL517413 0.71 CDK7 (0.54) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL29993829 0.71 CDK7 (0.54) CCNT1CCNKCDK9CDK12CCNE1
SCHEMBL28313446 0.71 PDE3B (0.42) AHRCDK1KDRULK1
SCHEMBL30957453 0.71 CHRM5 (0.46) CCNT1CCNKCDK9CDK12CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110036004-A Inhibitors of cyclin dependent kinase 7(CDK7) 希洛斯医药品股份有限公司 2019-07-19 CN disclosed