SCHEMBL28313446

SCHEMBL28313446

FC(F)(F)c1cnc(Cl)nc1-c1ccc2cc[nH]c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.42
PDE3A Q14432 2/20 0.42
AHR P35869 2/20 0.41
CMA1 P23946 1/20 0.41
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
RIPK2 O43353 1/20 0.39
KDR P35968 3/20 0.39
CDK1 P06493 2/20 0.39
MET P08581 1/20 0.39
MPO P05164 5/20 0.38
KCNH2 Q12809 2/20 0.38
PIK3CD O00329 1/20 0.38
ABL1 P00519 1/20 0.38
EGFR P00533 1/20 0.38
HCK P08631 1/20 0.38
SRC P12931 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
MTOR P42345 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29699016 0.73 NFKB1 (0.35) PIK3CDULK1
SCHEMBL29107848 0.71 AR (0.43) ADORA1ABL1EGFRSRC
SCHEMBL30578587 0.71 AR (0.43) ADORA1ABL1EGFRSRC
SCHEMBL27503715 0.71 NPC1 (0.41) ADORA2AADORA1
SCHEMBL28313382 0.71 AHR (0.44) AHRKDRCDK1ULK1
SCHEMBL4786964 0.70 AHR (0.49) AHRCMA1ADORA2AADORA1KDR
SCHEMBL14325223 0.69 AHR (0.41) AHRCMA1ADORA2AADORA1RIPK2
SCHEMBL24143483 0.69 TRPA1 (0.54) PDE3BPDE3AMPOKCNH2
SCHEMBL7091832 0.67 ESR1 (0.55) AHRCMA1METMPOKCNH2
SCHEMBL30837013 0.67 LRRK2 (0.47) KDRCDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110036004-A Inhibitors of cyclin dependent kinase 7(CDK7) 希洛斯医药品股份有限公司 2019-07-19 CN disclosed