SCHEMBL28313674

SCHEMBL28313674

CCONS(=O)(=O)c1cccnc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.49
NFE2L2 Q16236 1/20 0.49
LMNA P02545 1/20 0.48
NAPRT Q6XQN6 1/20 0.47
MAPT P10636 1/20 0.47
ALDH1A1 P00352 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
KMT2A Q03164 2/20 0.44
SLC40A1 Q9NP59 2/20 0.43
GLO1 Q04760 1/20 0.43
HIF1A Q16665 1/20 0.43
TSHR P16473 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 1/20 0.43
SLC1A3 P43003 1/20 0.43
SLC1A2 P43004 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3447394 0.80 ALDH1A1 (0.59) KEAP1NFE2L2LMNANAPRTMAPT
SCHEMBL2125283 0.79 KMT2A (0.50) KEAP1LMNAMAPTALDH1A1SMN1; SMN2
SCHEMBL16831885 0.77 SMN1; SMN2 (0.61) KEAP1NFE2L2LMNANAPRTMAPT
SCHEMBL6390027 0.76 HIF1A (0.50) KEAP1NFE2L2LMNANAPRTMAPT
SCHEMBL30338836 0.75 NAPRT (0.57) KEAP1NFE2L2NAPRTMAPTALDH1A1
SCHEMBL2227366 0.75 NAPRT (0.57) KEAP1NFE2L2NAPRTMAPTALDH1A1
SCHEMBL2371844 0.75 NAPRT (0.57) KEAP1NFE2L2NAPRTMAPTALDH1A1
SCHEMBL21960091 0.75 NAPRT (0.57) KEAP1NFE2L2LMNANAPRTMAPT
SCHEMBL18308968 0.75 TSHR (0.57) NAPRTMAPTALDH1A1SMN1; SMN2KMT2A
SCHEMBL28632022 0.75 NAPRT (0.52) KEAP1NFE2L2LMNANAPRTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110167946-A Sulfonamide compounds with TNAP inhibitory activity 第一三共株式会社 2019-08-23 CN disclosed