SCHEMBL28320196

SCHEMBL28320196

Nc1cccc(-c2ccc(NC=O)c3[nH]ncc23)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KIT P10721 1/20 0.39
NUDT1 P36639 1/20 0.36
METAP2 P50579 2/20 0.36
ENPP2 Q13822 1/20 0.36
PABPC1 P11940 1/20 0.36
ERBB2 P04626 1/20 0.36
TEC P42680 1/20 0.36
TXK P42681 1/20 0.36
BLK P51451 1/20 0.36
BMX P51813 1/20 0.36
JAK3 P52333 1/20 0.36
ITK Q08881 1/20 0.36
ERBB4 Q15303 1/20 0.36
NTRK1 P04629 3/20 0.35
PIK3CA P42336 1/20 0.35
GRK2 P25098 1/20 0.35
PDPK1 O15530 1/20 0.35
AURKA O14965 1/20 0.35
MAP4K4 O95819 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28321318 0.80 BTK (0.43) KITPABPC1
SCHEMBL28320237 0.78 BTK (0.54) JAK3ITKAURKA
SCHEMBL28321299 0.78 ASH1L (0.43) KITPABPC1
SCHEMBL28320214 0.76 KIT (0.35) KITPABPC1NTRK1PIK3CAMAP4K4
SCHEMBL28320183 0.76 KIT (0.39) KITNUDT1METAP2ENPP2ERBB2
SCHEMBL28321286 0.75 PARP1 (0.37) KITPABPC1
SCHEMBL16337236 0.75 BTK (0.50) ERBB2TECTXKBLKBMX
SCHEMBL28321282 0.74 TP53 (0.36) KITPABPC1NTRK1MAP4K4
SCHEMBL23518814 0.72 METAP2 (0.40) KITNUDT1METAP2ENPP2NTRK1
SCHEMBL28093874 0.70 METAP2 (0.68) KITMETAP2ENPP2ERBB2TEC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105530932-B Primary formamide as BTK inhibitor 艾伯维公司 2019-09-27 CN disclosed